G-protein/receptor inhibitors as blockers of receptor signaling

DOI10.1016/J.JTBI.2019.07.014zbMATH Open1420.92024OpenAlexW2965588471WikidataQ92253033 ScholiaQ92253033MaRDI QIDQ2324876FDOQ2324876

Authors: Terry Kenakin 

Publication date: 12 September 2019

Published in: Journal of Theoretical Biology (Search for Journal in Brave)

Full work available at URL: https://doi.org/10.1016/j.jtbi.2019.07.014

Recommendations

• Enhancer and competitive allosteric modulation model for G-protein-coupled receptors
• Kinetic operational models of agonism for G-protein-coupled receptors
• Mathematical modelling of signalling in a two-ligand G-protein coupled receptor system: agonist-antagonist competition
• Modelling of signalling via G-protein coupled receptors: pathway-dependent agonist potency and efficacy
• Modelling and simulation of biased agonism dynamics at a G protein-coupled receptor

zbMATH Keywords

allosteric antagonismG-protein receptor couplingreceptor antagonism

Mathematics Subject Classification ID

Biochemistry, molecular biology (92C40)

Cited In (1)

• Enhancer and competitive allosteric modulation model for G-protein-coupled receptors

This page was built for publication: G-protein/receptor inhibitors as blockers of receptor signaling

Report a bug (only for logged in users!)Click here to report a bug for this page (MaRDI item Q2324876)